<i>In vivo</i> evaluation of intestinal human CYP3A inhibition by macrolide antibiotics in CYP3A-humanised mice

نویسندگان

چکیده

Genki Minegishia, Yasuhiro Kazukibc, Shin-Ichiro Nittad, Atsushi Miyajimae, Hidetaka Akitaa & Kaoru Kobayashie*a Laboratory of DDS Design and Drug Disposition, Graduate School Pharmaceutical Sciences, Chiba University, Chiba, Japanb Chromosome Engineering Research Center (CERC), Tottori Tottori, Japanc Department Molecular Cellular Biology, Division Genome Functions, Faculty Medicine, Life Science, Japand Bioanalysis Department, Medical Solution Segment, Advanced Technology Center, LSI Medience Corporation, Tokyo, Japane Biopharmaceutics, Clinical Pharmacy, Meiji Japan

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ژورنال

عنوان ژورنال: Xenobiotica

سال: 2021

ISSN: ['1366-5928', '0049-8254']

DOI: https://doi.org/10.1080/00498254.2021.1921314